The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
Sinicropi, Maria
The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value - Basel, Switzerland MDPI - Multidisciplinary Digital Publishing Institute 2021 - 1 electronic resource (218 p.)
Open Access
The book explores issues concerning the design, synthetic methods and biological evaluation of molecules of pharmaceutical interest.
Creative Commons
English
books978-3-0365-1300-3 9783036512990 9783036513003
10.3390/books978-3-0365-1300-3 doi
Research & information: general
Chemistry
fluorinated pyrazole aldehydes tyrosinase inhibition phosphodiesterase inhibition antibacterial activity molecular docking periodontitis SRP LDD gelcide cancer phytocomponents Tiospora cardifolia silica silver oxynitrate stability core-shell antibiofilm antimicrobial sesquiterpene inflammatory pathologies nutraceuticals triclosan surgical site infection suture abdominal surgery cost-analysis budget impact analysis spirooxindole 1,3-dipolar cycloaddition eco-friendly chemistry ROCS shape alignment lipophilicity anticancer activity sol–gel coating medical textiles antioxidant anti-inflammatory PEA derivative drug release imidazole antiproliferative antioxidant activities docking DPPH ABTS acetylcholinesterase xanthine oxidase pyrimidine-trione barbituric thiobarbituric urease inhibitors DFT N-benzylisatin-aryl hydrazones gefitinib A549 cell lines pomegranate Punica granatum L. pomegranate skin extract pomegranate fruit extract nutraceutical properties biological properties cladodes Opuntia antioxidants polyphenols SFE-CO2 rutin iso-quercitrin nicotiflorin narcissin n/a
The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value - Basel, Switzerland MDPI - Multidisciplinary Digital Publishing Institute 2021 - 1 electronic resource (218 p.)
Open Access
The book explores issues concerning the design, synthetic methods and biological evaluation of molecules of pharmaceutical interest.
Creative Commons
English
books978-3-0365-1300-3 9783036512990 9783036513003
10.3390/books978-3-0365-1300-3 doi
Research & information: general
Chemistry
fluorinated pyrazole aldehydes tyrosinase inhibition phosphodiesterase inhibition antibacterial activity molecular docking periodontitis SRP LDD gelcide cancer phytocomponents Tiospora cardifolia silica silver oxynitrate stability core-shell antibiofilm antimicrobial sesquiterpene inflammatory pathologies nutraceuticals triclosan surgical site infection suture abdominal surgery cost-analysis budget impact analysis spirooxindole 1,3-dipolar cycloaddition eco-friendly chemistry ROCS shape alignment lipophilicity anticancer activity sol–gel coating medical textiles antioxidant anti-inflammatory PEA derivative drug release imidazole antiproliferative antioxidant activities docking DPPH ABTS acetylcholinesterase xanthine oxidase pyrimidine-trione barbituric thiobarbituric urease inhibitors DFT N-benzylisatin-aryl hydrazones gefitinib A549 cell lines pomegranate Punica granatum L. pomegranate skin extract pomegranate fruit extract nutraceutical properties biological properties cladodes Opuntia antioxidants polyphenols SFE-CO2 rutin iso-quercitrin nicotiflorin narcissin n/a
